姓名:李杰 职称:教授 部门:化学学院 联系方式: Email:jjackli@suda.edu.cn |
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01. 2020-至今教授,www.优德88.cpm‒材料与化学化工学部,苏州,江苏 10. 2017- 11.2019慕尼黑大学‒化学与药学院博士后研究员,慕尼黑,德国;(合作导师:Prof. Dr. Paul Knochel) 10. 2015- 10. 2017特聘研究员,江南大学‒药学院,无锡,江苏 08. 2015- 10. 2015访问学者,中国医学科学院药物研究所‒药物化学室(肖志艳研究员) 11. 2011- 07. 2015哥廷根大学‒有机化学与分子生物化学系博士,哥廷根,德国;(博士学位‒“summa cum laude”;合作导师:Prof. Dr. Lutz Ackermann). 08. 2009- 10. 2011中国医学科学院药物研究所‒药物化学室(硕士交换生;导师:肖志艳研究员). 09. 2008- 07. 2009沈阳药科大学‒(天然)药物化学系硕士(导师:华会明教授). 09. 2004- 06. 2008(学士学位).天津商业大学‒制药工程系 学历及学术经历:2012年至今以一作或通讯作者在J. Am. Chem. Soc., Angew. Chem. Int. Ed., ACS Catal., Org. Lett., Adv. Synth. Catal., Chem. Eur. J., J. Org. Chem.,等期刊上发表学术论文20余篇;入选2016年江苏省双创人才;目前完成国家自然科学基金青年项目一项、江苏省自然科学基金青年基金一项。
研究领域:
金属
有机化学
&
药物化学
代表性论文(*通讯作者):
1.Z. Zhang, L. Liu, Y. Wang, Y. Zhang,J. Li*,Electrophilic Amination with Anthranils through Cobalt(III)-Catalyzed C(sp3)‒H Activation.Synthesis2020,DOI: 10.1055/s-0039-1690087. 2.J. Li*, Q. Ren, X. Cheng, K. Karaghiosoff, P. Knochel*, Chromium(II)-Catalyzed Diastereoselective and Chemoselective Csp2‒Csp3Cross-Couplings Using Organomagnesium Reagents.J. Am. Chem. Soc.2019,141, 18127‒18135. 3.S. Han, S. Liu, L. Liu, L. Ackermann,J. Li*, Cobalt-Catalyzed Diastereoselective Difluoroalkyaltion/Giese Addition Domino Reactions.Org. Lett.2019,21, 5387‒5391. (Front Cover) 4.J. Li*, P. Knochel*, Chromium-Catalyzed Cross-Couplings and Related Reactions.Synthesis2019,51, 2100‒2106. 5.J. Li*, E. Tan, N. Keller, Y.-H. Chen, P. M. Zehetmaier, A. C. Jakowetz, T. Bein*, P. Knochel*, Cobalt-Catalyzed Electrophilic Amination with Anthranils: An Expedient Route to Condensed Quinolines.J. Am. Chem. Soc.2019,141, 98‒103.(highlighted inSynfact2019) 6.M. Tang, Y. Li,S. Han,L. Liu, L. Ackermann,J. Li*, Rhodium(III)-Catalyzed C‒H Alkylation/Nucleophilic Addition Domino Reaction.Eur. J. Org. Chem.2019, 660‒664. 7.Y. Da, S. Han, X. Du, S. Liu, L. Liu,J. Li*,Copper(I)-Catalyzed Oxydifluoroalkylation of Alkenes: A Route to Functionalization Lactones.Org. Lett.2018,20. 5149‒5152. 8.J. Li, P. Knochel*, Cobalt-Catalyzed Cross-Couplings between Alkenyl Acetates and Aryl or Alkenyl Zinc Pivalates.Angew. Chem. Int. Ed.2018,57, 11436‒11440. 9.Liang-Hua Zou*, Cong Zhao, Ping-Gui Li, Ying Wang,J. Li*,Transition-Metal-Free C−S Bond Formation: Synthesis of Polysubstituted Diaryl Sulfides and α‑Thioarylcarbonyl Compounds.J. Org. Chem.2017,82, 12892–12898. 10.X. Zhang*, H. Zheng,J. Li*, F. Xu, J. Zhao, H. Yan*, Selective Catalytic B–H Arylation ofo-Carboranyl Aldehydes by a Transient Directing Strategy.J. Am. Chem. Soc.2017,139, 14511‒14517. 11.Z. Zhang, S. Han, M. Tang, L. Ackermann*,J. Li*, C–H Alkylations of (Hetero)Arenes by Maleimides and Maleate Ester through Versatile Cobalt(III) Catalysis.Org. Lett.2017,19, 3135–3318. 12.S. Han, W. Ma, Z. Zhang, L. Liu, M. Tang,J. Li*, Mild C(sp3)‒H Alkylation of 8-Methylquinolines with α,β-Unsaturated Carbonyl Compounds by Rhodium(III) Catalysis.Asain J.Org. Chem.2017,6,1014‒1018.(Front Cover) 13.J. Li*, Z. Zhang, W. Ma, M. Tang, D. Wang, L.-H. Zou, Mild Cobalt(III)-Catalyzed C‒H Hydroarylation of Conjugated C=C/C=O Bonds.Adv. Synth. Catal.2017,359,1717–1724. 14.M. Moselage†,J. Li†(Co-first author), F. Kramm, L. Ackermann*, Ruthenium(II)-Catalyzed Decarbamoylative C–C Arylations and Alkylations.Angew. Chem. Int. Ed.2017,55, 5341–5344. 15.Z. Zhang, M. Tang, S. Han, L. Ackermann,J. Li*, Carboxylate Enhanced Rhodium(III)-Catalyzed ArylC–H Alkylation with Conjugated Alkenes under Mild Conditions.J. Org. Chem.2017,82, 664–672. 16.W. Ma*, P. Gandeepan*,J. Li, L. Ackermann*, Recent Advances in Positional-Selective Alkenylations: Removable Guidance for Twofold C‒H Activation.Org. Chem. Front.2017,4, 1435‒1467. 17.Z. Zhang, M. Tang, L. Zang, L.-H. Zou,J. Li*, Thermolysis of 2-Diazo-3-aryl ketoesters: New Route to α-Aryl Malonates and Aromatic Esters. Tetrahedron Lett.2016,57, 5681–5684. 18.J. Li*, Z. Zhang, M. Tang, X. Zhang, J. Jin,Selective Synthesis of Isoquinolines by Rhodium(III)-Catalyzed C–H/N–H Functionalization with α-Substituted Ketones. Org. Lett.2016,18, 3898–3901. 19.J. Li*, M. Tang, L. Zang, X. Zhang, Z. Zhang, L. Ackermann*,Amidines for Versatile Cobalt(III)-Catalyzed Synthesis of Isoquinolines through C–H Functionalization with Diazo Compounds. Org. Lett.2016,18, 2742–2745. (highlighted inOrganic Chemistry Portal2017) 20.M. Moselage†,J. Li†(Co-first author), L. Ackermann*, Cobalt-Catalyzed C–H Activation.ACS Catal.2016,6, 498–525. 21.J. Li, L. Ackermann*, Cobalt(III)-Catalyzed Aryl and Alkenyl C–H Aminocarbonylation with Isocyanates and Acyl Azides.Angew. Chem. Int. Ed.2015,54, 8551–8554. 22.J. Li, L. Ackermann*, Cobalt-Catalyzed C–H Cyanation of Arenes and Heteroarenes.Angew. Chem. Int. Ed.2015,54, 3635–3638. (Selected ashot paper,highlighted inChemCatChem2015,7, 732). 23.J. Li, L. Ackermann*, Cobalt-Catalyzed C–H Arylations with Weakly-Coordinating Amindes and Tetrazoles: Expedient Route to Angiotensin-II-Receptor Blockers.Chem. Eur. J.2015,21, 5718–5722. 24.J. Li, L. Ackermann*, Carboxylate-Assisted Ruthenium(II)-Catalyzed C–H Activations of Monodentate Amides with Conjugated Alkenes.Org. Chem. Front.2015,2, 1035–1039. 25.J. Li, M. John, L. Ackermann*, Amidines for Versatile Ruthenium(II)-Catalyzed Oxidative C–H Activations with Internal Alkynes and Acrylates.Chem. Eur. J.2014,20, 5403–5408. 26.J. Li,L. Ackermann*, Ruthenium-Catalyzed Oxidative Alkyne Annulation by C–H Activation on Ketimines.Tetrahedron2014,70, 3342–3348. 27.J. Li, H.-M. Hua, Y-B. Tang, S. Zhang, E. Ohkoshi, K.-H Lee, Z. Xiao*, Synthesis and Evaluation of Novel Podophyllotoxin Analogs.Bioorg. Med. Chem. Lett.2012,22, 4293–4295. |